This paper explores the medicinal uses, chemical properties, and methods of synthesis of organometallic compounds, highlighting their potential as therapeutic agents and their diverse reactivity. These compounds play a crucial role in treating diseases and metabolic disorders, with metal structures playing a kinetic role at the cellular level. The text emphasises the synthesis, mechanisms of action, and many therapeutic applications of these compounds, with a specific focus on their usage as anticancer agents, antibacterial agents, and in targeted drug administration. It seeks to investigate the wide array of organometallic compounds utilised in medicine, elucidating their methods of action as well as their present and prospective applications in the treatment of numerous ailments. This review seeks to offer a comprehensive examination of the therapeutic applications of organometallic compounds, encompassing their modes of operation, present uses, and potential advancements in the fields of drug development and treatment. However, the development of antiviral drugs cannot solely rely on organometallic complexes. Challenges include potential toxicity and the complexity of synthesis and characterization, which require specialized equipment and expertise.